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Synthesis of a boronic ester-appended bismuth(III) porphyrin as a potential alpha-particle bi-emitter

Université de Rennes 1, Sciences Chimiques de Rennes, UMR CNRS 6226 (I.C.M.V.), 35042 Rennes Cedex, France

Current address: Université Mentouri de Constantine, Laboratoire des produits naturels d'origine végétale et de synthèse organique, Département de Chimie, Faculté des Sciences, 25000 Constantine, Algérie

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Bertrand Carboni

Université de Rennes 1, Sciences Chimiques de Rennes, UMR CNRS 6226 (I.C.M.V.), 35042 Rennes Cedex, France

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Bernard Boitrel

Université de Rennes 1, Sciences Chimiques de Rennes, UMR CNRS 6226 (I.C.M.V.), 35042 Rennes Cedex, France

SPP full member in good standing

Corresponding author, fax: +33 (0)2 23 23 56 37

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https://doi.org/10.1142/S1088424608000030Cited by:7 (Source: Crossref)

Abstract

As ²¹³Bi, a spontaneous alpha-emitting radioisotope, and ¹⁰B, a neutron-activated source of alpha particles, have been found to be potential tools in the treatment of cancer patients, a novel bismuth porphyrin, bearing both boron atoms and a strap with a hanging carboxylic group, was synthesized.

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